Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04706
Ion Channel
Sodium channel protein type 2 subunit alpha
Peptide Function
Blocker
Gene Name
SCN2A
Activity Data (nM)
IC50
Not available
Ki
Not available
EC50
Not available
Kd
5.3 nM
Biologically Active
Not specified
Sequence Information
Peptide Sequence
CCNCSSKWCRDHSRCC
Peptide UniProt Accession
UniParc
UPI0000603521
Peptide Synonyms/Alias
[mu-Conotoxin K IIIA; UNII-390H5GUO40; CHEMBL2402969; 390H5GUO40; 884469-67-4; Ccncsskwcrdhsrcc-NH2 cyclic (1->9);(2->15);(4->16); L-Cysteinamide; L-cysteinyl-L-cysteinyl-L-asparaginyl-L-cysteinyl-L-seryl-L-seryl-L-lysyl-L-tryptophyl-L-cysteinyl-L-arginyl-L-alpha-aspartyl-L-histidyl-L-seryl-L-arginyl-L-cysteinyl-; cyclic (1->9);(2->15);(4->16)-tris(disulfide); mu-Conotoxin KIIIA; BDBM50492340; DA-68915]
Peptide Species
Conus kinoshitai
Peptide Name
Mu-conotoxin KIIIB
CAS Number
884469-67-4
Experimental Conditions
pH
pH 7.5
Holding Potential (mV)
−80 mV
Temperature
20 ℃
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available